Clopidogrel resistance is associated with increased risk of recurrent atherothrombotic events in patients with acute myocardial infarction

Circulation. 2004 Jun 29;109(25):3171-5. doi: 10.1161/01.CIR.0000130846.46168.03. Epub 2004 Jun 7.

Abstract

Background: Although clopidogrel reduces the risk of cardiovascular episodes after coronary events and stenting, a substantial number of incidents continue to occur.

Methods and results: The antiplatelet effect of clopidogrel was studied prospectively in 60 consecutive patients who underwent primary angioplasty (percutaneous coronary intervention [PCI]) with stenting for acute ST-segment-elevation myocardial infarction (STEMI) to determine whether variability in response to clopidogrel affects clinical outcomes. Patients were stratified into 4 quartiles according to the percentage reduction of ADP-induced platelet aggregation. Although patients in the first quartile were resistant to the effects of clopidogrel (ADP-induced platelet aggregation at day 6, 103+/-8% of baseline), ADP-induced aggregation was reduced to 69+/-3%, 58+/-7%, and 33+/-12% of baseline, respectively, in patients in quartiles 2 through 4 (P<0.01 for all). In addition, epinephrine-induced platelet aggregation and platelet aggregation under flow conditions, assessed by the cone-and-plate(let) analyzer method, were reduced significantly less in the first quartile than in quartiles 2 through 4. Whereas 40% of patients in the first quartile sustained a recurrent cardiovascular event during a 6-month follow-up, only 1 patient (6.7%) in the second quartile and none in the third and fourth quartiles suffered a cardiovascular event (P=0.007).

Conclusions: Up to 25% of STEMI patients undergoing primary PCI with stenting are resistant to clopidogrel and therefore may be at increased risk for recurrent cardiovascular events.

Publication types

  • Comparative Study

MeSH terms

  • Adenosine Diphosphate / antagonists & inhibitors
  • Adenosine Diphosphate / pharmacology
  • Aged
  • Aspirin / administration & dosage
  • Aspirin / therapeutic use
  • Biotransformation
  • Clopidogrel
  • Combined Modality Therapy
  • Coronary Artery Disease / complications*
  • Coronary Artery Disease / therapy
  • Coronary Restenosis / epidemiology*
  • Coronary Restenosis / prevention & control
  • Coronary Thrombosis / epidemiology
  • Coronary Thrombosis / etiology
  • Coronary Thrombosis / prevention & control
  • Drug Resistance
  • Drug Therapy, Combination
  • Epinephrine / administration & dosage
  • Epinephrine / therapeutic use
  • Eptifibatide
  • Female
  • Follow-Up Studies
  • Humans
  • Male
  • Middle Aged
  • Myocardial Infarction / drug therapy*
  • Myocardial Infarction / etiology
  • Myocardial Infarction / prevention & control
  • Myocardial Infarction / therapy
  • Peptides / therapeutic use
  • Platelet Aggregation / drug effects
  • Platelet Aggregation Inhibitors / pharmacology*
  • Platelet Aggregation Inhibitors / therapeutic use
  • Prodrugs / pharmacology*
  • Prodrugs / therapeutic use
  • Prospective Studies
  • Purinergic P2 Receptor Antagonists
  • Recurrence
  • Risk
  • Smoking / epidemiology
  • Stents
  • Ticlopidine / analogs & derivatives*
  • Ticlopidine / pharmacology*
  • Ticlopidine / therapeutic use
  • Treatment Outcome

Substances

  • Peptides
  • Platelet Aggregation Inhibitors
  • Prodrugs
  • Purinergic P2 Receptor Antagonists
  • Adenosine Diphosphate
  • Clopidogrel
  • Eptifibatide
  • Ticlopidine
  • Aspirin
  • Epinephrine