Practical synthesis of new and highly efficient ligands for the Suzuki reaction of aryl chlorides

Chem Commun (Camb). 2004 Jan 7:(1):38-9. doi: 10.1039/b311268n. Epub 2003 Nov 28.

Abstract

A practical synthesis of a novel class of phosphine ligands, phosphino substituted N-aryl pyrroles (PAP ligands), has been developed. These ligands are applied in the palladium-catalyzed coupling of a variety of aryl and heteroaryl chlorides with phenylboronic acid showing exceedingly high turnover numbers at mild reaction temperatures and even at room temperature.