TRPV4 calcium entry channel: a paradigm for gating diversity

Am J Physiol Cell Physiol. 2004 Feb;286(2):C195-205. doi: 10.1152/ajpcell.00365.2003.

Abstract

The vanilloid receptor-1 (VR1, now TRPV1) was the founding member of a subgroup of cation channels within the TRP family. The TRPV subgroup contains six mammalian members, which all function as Ca2+ entry channels gated by a variety of physical and chemical stimuli. TRPV4, which displays 45% sequence identity with TRPV1, is characterized by a surprising gating promiscuity: it is activated by hypotonic cell swelling, heat, synthetic 4alpha-phorbols, and several endogenous substances including arachidonic acid (AA), the endocannabinoids anandamide and 2-AG, and cytochrome P-450 metabolites of AA, such as epoxyeicosatrienoic acids. This review summarizes data on TRPV4 as a paradigm of gating diversity in this subfamily of Ca2+ entry channels.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Amino Acid Sequence / genetics
  • Animals
  • Calcium / metabolism
  • Cation Transport Proteins / agonists
  • Cation Transport Proteins / genetics
  • Cation Transport Proteins / metabolism*
  • Cation Transport Proteins / physiology
  • Gene Expression
  • Hot Temperature
  • Humans
  • Ion Channel Gating / physiology*
  • Ion Channels / agonists
  • Ion Channels / genetics
  • Ion Channels / metabolism*
  • Ion Channels / physiology
  • Mechanoreceptors / physiology
  • Molecular Sequence Data
  • Osmotic Pressure
  • Phosphorylation
  • TRPV Cation Channels

Substances

  • Cation Transport Proteins
  • Ion Channels
  • TRPV Cation Channels
  • TRPV4 protein, human
  • Calcium