A novel strategy towards the synthesis of orthogonally functionalised 4-aminoglycosides

Org Biomol Chem. 2003 Dec 7;1(23):4160-5. doi: 10.1039/b309823k. Epub 2003 Oct 21.

Abstract

A tethered nucleophilic substitution strategy for the stereoselective introduction of axially oriented amino functions on suitably protected gluco- and mannopyranosides is presented. The obtained oxazine is a versatile building block, which after some manipulation, could be used in the construction of highly functionalised oligosaccharides.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aminoglycosides / chemical synthesis*
  • Aminoglycosides / chemistry*
  • Molecular Structure
  • Stereoisomerism

Substances

  • Aminoglycosides