Stimulation of postsynaptic 5-HT1A receptors is responsible for the anticonflict effect of ipsapirone in rats

J Pharm Pharmacol. 1992 Sep;44(9):780-2. doi: 10.1111/j.2042-7158.1992.tb05521.x.

Abstract

Ipsapirone (1.25-10 mg kg-1), a non-benzodiazepine anxiolytic drug with high affinity for 5-hydroxytryptamine1A (5-HT1A) receptors, increased dose-dependently the number of punished licks in the drinking conflict test (Vogel test) in rats. The anticonflict effect of the drug administered at a dose of 5 mg kg-1 was not modified in animals with lesions of 5-HT neurones, produced by p-chloroamphetamine (PCA, 2 x 10 mg kg-1). The anticonflict effect of ipsapirone in PCA-pretreated rats was antagonized by the 5-HT1A receptor and alpha 1-adrenoceptor antagonist NAN-190 (1-(2-methoxyphenyl)-4-[4-(2-phthalimmido)]butylpiperazine hydrobromide; 0.5-1 mg kg-1), but not by the selective alpha 1-adrenoceptor blocker prazosin (0.5 mg kg-1). Neither NAN-190 nor prazosin affected the punished response in PCA-pretreated rats. The present results indicate that the anticonflict effect of ipsapirone depends on stimulation of postsynaptic 5-HT1A receptors.

MeSH terms

  • Animals
  • Anti-Anxiety Agents / pharmacology*
  • Brain Chemistry / drug effects
  • Conflict, Psychological*
  • Male
  • Piperazines / pharmacology
  • Pyrimidines / pharmacology*
  • Rats
  • Rats, Wistar
  • Receptors, Serotonin / drug effects
  • Receptors, Serotonin / metabolism*
  • Serotonin Antagonists / pharmacology
  • p-Chloroamphetamine / pharmacology

Substances

  • Anti-Anxiety Agents
  • Piperazines
  • Pyrimidines
  • Receptors, Serotonin
  • Serotonin Antagonists
  • 1-(2-methoxyphenyl)-4-(4-(2-phthalimido)butyl)piperazine
  • p-Chloroamphetamine
  • ipsapirone