2'-modified-2-thiothymidine oligonucleotides

Org Lett. 2003 Aug 21;5(17):3005-8. doi: 10.1021/ol0348607.

Abstract

[reaction: see text] Oligonucleotides with novel modifications, 2'-O-[2-(methoxy)ethyl]-2-thiothymidine and 2'-deoxy-2'-fluoro-2-thiothymidine, have been synthesized. These modified oligonucleotides exhibited very high thermal stability when hybridized with complementary RNA. 2-O-(2-Methoxy)ethyl-2-thiothymidine modified oligonucleotide phosphodiesters showed enhanced resistance toward nucleases (t(1/2) > 24 h), but 2'-deoxy-2'-fluoro-2-thiothymidine modified oligonucleotide phosphodiesters showed limited stability to nucleotytic degradation.

MeSH terms

  • Animals
  • Base Sequence
  • DNA, Complementary / chemistry
  • Drug Stability
  • Hot Temperature
  • Oligonucleotides / chemical synthesis*
  • Oligonucleotides / chemistry
  • Oligonucleotides / metabolism
  • Phosphoric Diester Hydrolases / metabolism
  • RNA, Complementary / chemistry
  • Snake Venoms
  • Thymidine / analogs & derivatives*

Substances

  • DNA, Complementary
  • Oligonucleotides
  • RNA, Complementary
  • Snake Venoms
  • Phosphoric Diester Hydrolases
  • Thymidine