Suprachiasmatic nucleus circadian oscillatory protein, a novel binding partner of K-Ras in the membrane rafts, negatively regulates MAPK pathway

J Biol Chem. 2003 Apr 25;278(17):14920-5. doi: 10.1074/jbc.M213214200. Epub 2003 Feb 19.

Abstract

Suprachiasmatic nucleus circadian oscillatory protein (SCOP) is a member of the leucine-rich repeat (LRR)-containing protein family. In addition to circadian expression in the rat hypothalamic suprachiasmatic nucleus, SCOP is constitutively expressed in neurons throughout the rat brain. Here we found that a substantial amount of SCOP was localized in the brain membrane rafts, in which only K-Ras was abundant among Ras isoforms. SCOP interacted directly through its LRR domain with a subset of K-Ras in the guanine nucleotide-free form that was present in the raft fraction. This interaction interfered with the binding of added guanine nucleotide to K-Ras in vitro. A negative regulatory role of SCOP for K-Ras function was examined in PC12 cell lines stably overexpressing SCOP or its deletion mutants. Overexpression of full-length SCOP markedly down-regulated ERK1/ERK2 activation induced by depolarization or phorbol ester stimulation, and this inhibitory effect of overexpressed SCOP was dependent on its LRR domain. These results strongly suggest that SCOP negatively regulates K-Ras signaling in the membrane rafts, identifying a novel mechanism for regulation of the Ras-MAPK pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Down-Regulation
  • Guanosine Triphosphate / metabolism
  • MAP Kinase Signaling System*
  • Male
  • Membrane Microdomains / chemistry*
  • Mitogen-Activated Protein Kinases / metabolism
  • Mutation
  • Nuclear Proteins / genetics
  • Nuclear Proteins / metabolism*
  • Nuclear Proteins / physiology
  • PC12 Cells
  • Phosphoprotein Phosphatases
  • Phosphorylation
  • Protein Binding
  • Rats
  • Transfection
  • ras Proteins / metabolism*

Substances

  • Nuclear Proteins
  • Guanosine Triphosphate
  • Mitogen-Activated Protein Kinases
  • PHLPP1 protein, rat
  • Phosphoprotein Phosphatases
  • ras Proteins