Response of Apc(min) and A33 (delta N beta-cat) mutant mice to treatment with tea, sulindac, and 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine (PhIP)

Mutat Res. 2002 Sep 30:506-507:121-7. doi: 10.1016/s0027-5107(02)00158-6.

Abstract

There is growing interest in the potential health benefits of tea, and a recent report described the potent antimutagenic activity of white tea in comparison with green tea against several heterocyclic amines, including 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine (PhIP) [Mutat. Res. 495 (2001) 61]. We compared the inhibitory effects of white and green teas with sulindac, a nonsteroidal anti-inflammatory agent, in two different mouse models of intestinal tumorigenesis. In the Apc(min) mouse, white and green teas given at human-relevant concentrations (1.5% w/v, 2-min brew), and sulindac (80 ppm in the drinking water), each suppressed polyp formation by approximately 50%, and the combination of white tea plus sulindac was more effective than either treatment alone (P=0.05). Mice expressing an N-terminally truncated, oncogenic version of beta-catenin (A 33(delta N beta-cat) mutant mice) developed colonic aberrant crypt foci (ACF) spontaneously, but PhIP treatment increased the incidence and number of ACF per colon. In the normal-looking intestinal mucosa of Apc(min) and A 33(delta N beta-cat) mice, white tea plus sulindac treatment markedly attenuated the expression of beta-catenin protein, and this was recapitulated in vitro in cells transiently transfected with beta-catenin plus Tcf-4 and treated with tea or the major tea polyphenol epigallocatechin-3-gallate (EGCG). Expression of a beta-catenin/Tcf reporter was inhibited by EGCG in the transfected cells, and the beta-catenin/Tcf target genes cyclin D1 and c-jun were downregulated in vivo by tea plus sulindac treatment. Collectively, the data support a chemopreventive role for tea and sulindac against intermediate and late stages of colon cancer, via effects on the beta-catenin/Tcf signaling pathway.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenomatous Polyposis Coli Protein / deficiency
  • Adenomatous Polyposis Coli Protein / genetics
  • Adenomatous Polyposis Coli Protein / metabolism*
  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Catechin / analogs & derivatives*
  • Catechin / pharmacology
  • Cell Line
  • Cytoskeletal Proteins / deficiency
  • Cytoskeletal Proteins / genetics
  • Cytoskeletal Proteins / metabolism
  • Drug Combinations
  • Imidazoles / toxicity
  • Intestinal Mucosa / drug effects
  • Intestinal Mucosa / metabolism
  • Intestinal Neoplasms / chemically induced
  • Intestinal Neoplasms / metabolism
  • Intestinal Neoplasms / prevention & control*
  • Luciferases / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Mutant Strains
  • Plant Extracts / pharmacology*
  • Polyps / chemically induced
  • Polyps / metabolism
  • Polyps / prevention & control*
  • Sulindac / pharmacology*
  • Tea*
  • Trans-Activators / deficiency
  • Trans-Activators / genetics
  • Trans-Activators / metabolism
  • beta Catenin

Substances

  • Adenomatous Polyposis Coli Protein
  • Anti-Inflammatory Agents, Non-Steroidal
  • CTNNB1 protein, mouse
  • Cytoskeletal Proteins
  • Drug Combinations
  • Imidazoles
  • Plant Extracts
  • Tea
  • Trans-Activators
  • beta Catenin
  • Sulindac
  • Catechin
  • 2-amino-1-methyl-6-phenylimidazo(4,5-b)pyridine
  • epigallocatechin gallate
  • Luciferases