[8-chloroadenosine inhibits the growth factor-induced proliferation of retinal pigment epithelial cells in vitro]

Zhonghua Yan Ke Za Zhi. 1998 Jul;34(4):270-2.
[Article in Chinese]

Abstract

Objective: To study the inhibitory effect of 8-chloroadenosine (8-Cl-A) on growth factor-induced proliferation of retinal pigment epithelial (RPE) cells in vitro.

Methods: Primary culture and subculture of bovine RPE cells were established in vitro first and then tumor necrosis factor-alpha (TNF-alpha), interleukin-1beta (IL-1beta), basic fibroblast growth factor (bFGF) plus different concentrations of 8-Cl-A (2-16 micromol/L) were added to the cells of third passage respectively. DNA synthesis in RPE cells was measured with (3)H-TdR incorporation.

Results: Cells treated with TNF-alpha, IL-1beta, bFGF had a higher (3)H-TdR uptake than the basal. The increase was abolished by 8-Cl-A in a dose dependent manner (P < 0.05). At TNF-alpha, IL-1beta, bFGF with 8-Cl-A group, CPM was similar to basal at 16, 8, 2 micromol/L respectively (P > 0.05).

Conclusion: 8-Cl-A can inhibit the three growth factor-induced proliferation of RPE cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 2-Chloroadenosine / analogs & derivatives*
  • 2-Chloroadenosine / pharmacology*
  • Animals
  • Cattle
  • Cell Division / drug effects
  • DNA / biosynthesis
  • Dose-Response Relationship, Drug
  • Fibroblast Growth Factor 2 / antagonists & inhibitors
  • Interleukin-1 / antagonists & inhibitors
  • Pigment Epithelium of Eye / cytology
  • Pigment Epithelium of Eye / drug effects*
  • Tumor Necrosis Factor-alpha / antagonists & inhibitors

Substances

  • Interleukin-1
  • Tumor Necrosis Factor-alpha
  • Fibroblast Growth Factor 2
  • 2-Chloroadenosine
  • DNA
  • 8-chloroadenosine