Hepatitis C virus replication is directly inhibited by IFN-alpha in a full-length binary expression system

Proc Natl Acad Sci U S A. 2001 Aug 14;98(17):9847-52. doi: 10.1073/pnas.171319698. Epub 2001 Aug 7.

Abstract

Hepatitis C virus (HCV) is a leading cause of chronic hepatitis, cirrhosis, and hepatocellular carcinoma. The absence of culture systems permissive for HCV replication has presented a major bottleneck to antiviral development. We sought to recapitulate the early steps in the life cycle of HCV by means of DNA-based expression of viral genomic sequences. Here we report expression of replicating HCV RNA by using a, to our knowledge, novel binary expression system in which cells were transfected with a T7 polymerase-driven full-length HCV cDNA plasmid containing a cis-acting hepatitis Delta ribozyme to control 3' cleavage, and infected with vaccinia-T7 polymerase. HCV genomic and replicative strand synthesis, in addition to protein synthesis, was detectable and depended on full-length HCV sequences. Moreover, the system was capable of generating HCV RNA quasispecies, consistent with the action of the low-fidelity HCV NS5B RNA polymerase. IFN-alpha, but not ribavirin, directly inhibited the viral replicative cycle in these cells, identifying the virus itself and not solely the immune system as a direct target of IFN action. The availability of a cell-based test for viral replication will facilitate screening of inhibitory compounds, analysis of IFN-resistance mechanisms, and analysis of virus-host cell interactions.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amantadine / pharmacology
  • Animals
  • Antiviral Agents / pharmacology*
  • Bacteriophage T7 / genetics
  • Carcinoma, Hepatocellular / pathology
  • Chlorocebus aethiops
  • DNA, Complementary / genetics
  • Gene Expression Regulation, Viral / drug effects*
  • Genes, Synthetic
  • Hepacivirus / drug effects*
  • Hepacivirus / physiology
  • Humans
  • Interferon-alpha / pharmacology*
  • Liver Neoplasms / pathology
  • Oligodeoxyribonucleotides, Antisense / chemical synthesis
  • Oligodeoxyribonucleotides, Antisense / genetics
  • Polymerase Chain Reaction
  • RNA, Catalytic / genetics
  • RNA, Viral / biosynthesis
  • Reverse Transcriptase Polymerase Chain Reaction
  • Ribavirin / pharmacology
  • Terminator Regions, Genetic
  • Transfection
  • Tumor Cells, Cultured
  • Viral Proteins / biosynthesis
  • Viral Proteins / genetics
  • Virus Replication / drug effects*

Substances

  • Antiviral Agents
  • DNA, Complementary
  • Interferon-alpha
  • Oligodeoxyribonucleotides, Antisense
  • RNA, Catalytic
  • RNA, Viral
  • Viral Proteins
  • Ribavirin
  • Amantadine