Comparative evaluation of fecal fat excretion induced by orlistat and chitosan

Obes Res. 2001 Jun;9(6):364-7. doi: 10.1038/oby.2001.47.

Abstract

Objective: To compare the effects of chitosan and orlistat on fecal fat excretion.

Research methods and procedure: A randomized, open-label, two-period sequential design study was used. A total of 12 healthy adult volunteers within 20% of their ideal body weight entered a 7-day run-in diet period before being randomized to orlistat (120 mg) or chitosan (890 mg) three times daily for 7 days. Subjects then crossed over treatment regimens for an additional 7-day period. Subjects followed a standardized diet (2500 kcal/d, 30% as fat) for the entire 21-day study. Feces were collected on days 4 to 7 of the run-in period (baseline) and during the two treatment periods. Mean daily fecal fat excretion was measured at baseline and during each treatment regimen.

Results: Mean baseline fecal fat excretion for all subjects was 1.36 +/- 0.45 g/d. During orlistat treatment, mean fecal fat excretion significantly increased from baseline (+16.13 +/- 7.27 g/d; p < 0.001). No significant effect was observed with chitosan (+0.27 +/- 1.02 g/d; p = 0.379). Fecal fat excretion was significantly greater with orlistat than with chitosan (p < 0.001; 95% confidence intervals: 11.73; 20.00 g/d).

Discussion: This study provides additional evidence of the inhibitory effect of orlistat on dietary fat absorption. Chitosan, however, has no effect on fecal fat excretion.

Publication types

  • Clinical Trial
  • Comparative Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Anti-Obesity Agents / pharmacology*
  • Anticholesteremic Agents / pharmacology*
  • Chitin / analogs & derivatives
  • Chitin / pharmacology*
  • Chitosan
  • Dietary Fats / pharmacokinetics*
  • Feces / chemistry*
  • Female
  • Humans
  • Intestinal Absorption / drug effects
  • Lactones / pharmacology*
  • Lipids / analysis
  • Male
  • Middle Aged
  • Orlistat

Substances

  • Anti-Obesity Agents
  • Anticholesteremic Agents
  • Dietary Fats
  • Lactones
  • Lipids
  • Chitin
  • Chitosan
  • Orlistat