Activated MEK5 induces serial assembly of sarcomeres and eccentric cardiac hypertrophy

EMBO J. 2001 Jun 1;20(11):2757-67. doi: 10.1093/emboj/20.11.2757.

Abstract

Mitogen-activated protein kinase (MAPK) pathways couple intrinsic and extrinsic signals to hypertrophic growth of cardiomyocytes. The MAPK kinase MEK5 activates the MAPK ERK5. To investigate the potential involvement of MEK5-ERK5 in cardiac hypertrophy, we expressed constitutively active and dominant-negative forms of MEK5 in cardiomyocytes in vitro. MEK5 induced a form of hypertrophy in which cardiomyocytes acquired an elongated morphology and sarcomeres were assembled in a serial manner. The cytokine leukemia inhibitory factor (LIF), which stimulates MEK5 activity, evoked a similar response. Moreover, a dominant-negative MEK5 mutant specifically blocked LIF-induced elongation of cardiomyocytes and reduced expression of fetal cardiac genes without blocking other aspects of LIF-induced hypertrophy. Consistent with the ability of MEK5 to induce serial assembly of sarcomeres in vitro, cardiac-specific expression of activated MEK5 in transgenic mice resulted in eccentric cardiac hypertrophy that progressed to dilated cardiomyopathy and sudden death. These findings reveal a specific role for MEK5-ERK5 in the induction of eccentric cardiac hypertrophy and in transduction of cytokine signals that regulate serial sarcomere assembly.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Animals, Newborn
  • Apoptosis
  • COS Cells
  • Cardiomyopathy, Dilated / genetics
  • Cardiomyopathy, Dilated / pathology
  • Cardiomyopathy, Dilated / physiopathology*
  • Cells, Cultured
  • Chlorocebus aethiops
  • Enzyme Activation
  • Growth Inhibitors / pharmacology
  • Heart / physiopathology*
  • Heart Ventricles
  • Humans
  • Interleukin-6*
  • Leukemia Inhibitory Factor
  • Lymphokines / pharmacology
  • MAP Kinase Kinase 5
  • Mice
  • Mice, Transgenic
  • Mitogen-Activated Protein Kinase 7
  • Mitogen-Activated Protein Kinase Kinases / genetics
  • Mitogen-Activated Protein Kinase Kinases / metabolism*
  • Mitogen-Activated Protein Kinases / metabolism*
  • Myocardium / cytology
  • Myocardium / enzymology*
  • Myocardium / pathology
  • Rats
  • Recombinant Proteins / metabolism
  • Sarcomeres / physiology*
  • Sequence Deletion
  • Transfection

Substances

  • Growth Inhibitors
  • Interleukin-6
  • LIF protein, human
  • Leukemia Inhibitory Factor
  • Lif protein, mouse
  • Lymphokines
  • Recombinant Proteins
  • Mitogen-Activated Protein Kinase 7
  • Mitogen-Activated Protein Kinases
  • MAP Kinase Kinase 5
  • MAP2K5 protein, human
  • Map2k5 protein, rat
  • Mitogen-Activated Protein Kinase Kinases