Chromosomes 4 and 13 in beta-carboline-induced seizures in mice: benzodiazepine binding

Neuroreport. 2000 Jul 14;11(10):2157-61. doi: 10.1097/00001756-200007140-00019.

Abstract

Methyl beta-carboline-3-carboxylate (beta-CCM) is a ligand for the benzodiazepine (BZD) binding site of the GABA-A receptors with convulsive properties. We provided evidence for the involvement of a fragment of mouse chromosomes 4 and 13 in beta-CCM-induced seizures in a previous paper. Here, we analyzed, through [3H]-flumazenil binding, whether central BZD binding sites could be involved in the physiological processes underlying these differences of genetic sensitivities. In the JE/Le strain, where the effects of the chromosome 4 fragment can be analyzed, we found associations between [3H]-flumazenil binding and the convulsive action of beta-CCM. On the contrary, this no longer holds true in C3XtEso strain, where the effects of the chromosome 13 fragment were observed.

MeSH terms

  • Animals
  • Brain / drug effects
  • Brain / metabolism*
  • Carbolines / pharmacology*
  • Chromosome Mapping*
  • Convulsants / pharmacology*
  • Flumazenil / pharmacokinetics
  • Mice
  • Mice, Inbred Strains
  • Mice, Mutant Strains
  • Radioligand Assay
  • Receptors, GABA-A / drug effects
  • Receptors, GABA-A / physiology*
  • Seizures / chemically induced
  • Seizures / genetics*
  • Seizures / physiopathology
  • Species Specificity
  • Tritium

Substances

  • Carbolines
  • Convulsants
  • Receptors, GABA-A
  • Tritium
  • Flumazenil
  • beta-carboline-3-carboxylic acid methyl ester