Ca(2+) entry activated by S-nitrosylation. Relationship to store-operated ca(2+) entry

J Biol Chem. 1999 Dec 10;274(50):35318-24. doi: 10.1074/jbc.274.50.35318.

Abstract

The coupling between Ca(2+) pools and store-operated Ca(2+) entry channels (SOCs) remains an unresolved question. Recently, we revealed that Ca(2+) entry could be activated in response to S-nitrosylation and that this process was stimulated by Ca(2+) pool emptying (Favre, C. J., Ufret-Vincenty, C. A., Stone, M. R., Ma, H-T. , and Gill, D. L. (1998) J. Biol. Chem. 273, 30855-30858). In DDT(1)MF-2 smooth muscle cells and DC-3F fibroblasts, Ca(2+) entry activated by the lipophilic NO donor, GEA3162 (5-amino-3-(3, 4-dichlorophenyl)1,2,3,4-oxatriazolium), or the alkylator, N-ethylmaleimide, was observed to be strongly activated by transient external Ca(2+) removal, closely resembling activation of SOC activity in the same cells. The nonadditivity of SOC and NO donor-activated Ca(2+) entry suggested a single entry mechanism. Calyculin A-induced reorganization of the actin cytoskeleton prevented SOC but had no effect on GEA3162-induced Ca(2+) entry. However, a single entry mechanism could account for both SOC and NO donor-activated entry if the latter reflected direct modification of the entry channel by S-nitrosylation, bypassing the normal coupling process between channels and pools. Small differences between SOC and GEA3162-activated Ba(2+) entry and sensitivity to blockade by La(3+) were observed, and in HEK293 cells SOC activity was observed without a response to thiol modification. It is concluded that in some cells, S-nitrosylation modifies an entry mechanism closely related to SOC and/or part of the regulatory machinery for SOC-mediated Ca(2+) entry.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Barium / pharmacokinetics
  • Calcium / metabolism*
  • Calcium Channels / drug effects
  • Calcium Channels / physiology*
  • Cell Line
  • Cricetinae
  • Ethylmaleimide / pharmacology
  • Kinetics
  • Muscle, Smooth
  • Nitric Oxide Donors / pharmacology*
  • Nitroso Compounds
  • Platelet Aggregation Inhibitors / pharmacology
  • Thapsigargin / pharmacology
  • Triazoles / pharmacology*

Substances

  • Calcium Channels
  • Nitric Oxide Donors
  • Nitroso Compounds
  • Platelet Aggregation Inhibitors
  • Triazoles
  • Barium
  • Thapsigargin
  • GEA 3162
  • Ethylmaleimide
  • Calcium