Effects of low-dose monophasic levonorgestrel with ethinyl estradiol preparation on serum lipid levels: A twenty-four month clinical trial

Am J Obstet Gynecol. 1999 Nov;181(5 Pt 2):59-62. doi: 10.1016/s0002-9378(99)70365-0.

Abstract

Objective: The aim of this 24-cycle study was to evaluate the effects on serum lipid concentrations of an oral contraceptive preparation containing 100 microg levonorgestrel and 20 microg ethinyl estradiol.

Study design: Forty-two healthy women were enrolled in a study designed to evaluate the effects on serum lipid concentrations of an oral contraceptive containing 100 microg levonorgestrel and 20 microg ethinyl estradiol. Lipid data were evaluated for 28 women who completed 24 cycles of treatment with a preparation of 100 microg levonorgestrel with 20 microg ethinyl estradiol for 21 days followed by placebo for 7 days. Concentrations of triglycerides, total cholesterol, high-density lipoprotein cholesterol, high-density lipoprotein cholesterol subfractions 2 and 3, low-density lipoprotein cholesterol, and apolipoproteins A-I and B were analyzed. Mean percentage changes from baseline were tested for significance by means of paired Student t tests.

Results: Total cholesterol, high-density lipoprotein cholesterol, high-density lipoprotein subfraction 2, and apolipoprotein A-I concentrations were not significantly changed from baseline. Neither was the ratio of high-density lipoprotein subfraction 2 to high-density lipoprotein subfraction 3. Mean percentage increases in concentrations of triglyceride, high-density lipoprotein subfraction 3, apolipoprotein B, and low-density lipoprotein cholesterol and increases in the ratios of total cholesterol to high-density lipoprotein cholesterol, low-density lipoprotein cholesterol to high-density lipoprotein cholesterol, and apolipoprotein B to apolipoprotein A-I were significant (P <.05) at >/=1 cycle. By cycle 24, however, only the concentration of high-density lipoprotein subfraction 3 remained significantly elevated.

Conclusion: Changes in the plasma lipid profiles among women receiving monophasic 100 microg levonorgestrel with 20 microg ethinyl estradiol were similar to those seen with other low-dose oral contraceptives, but by cycle 24 only 1 of 7 mean values remained significantly different from baseline.

Publication types

  • Clinical Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Contraceptive Agents, Female / administration & dosage*
  • Contraceptive Agents, Female / therapeutic use
  • Contraceptives, Oral, Synthetic / administration & dosage*
  • Contraceptives, Oral, Synthetic / therapeutic use
  • Dose-Response Relationship, Drug
  • Drug Combinations
  • Estradiol Congeners / administration & dosage*
  • Estradiol Congeners / therapeutic use
  • Ethinyl Estradiol / administration & dosage*
  • Ethinyl Estradiol / therapeutic use
  • Female
  • Humans
  • Levonorgestrel / administration & dosage*
  • Levonorgestrel / therapeutic use
  • Lipids / blood*
  • Lipoproteins, HDL / blood
  • Lipoproteins, LDL / blood
  • Longitudinal Studies

Substances

  • Contraceptive Agents, Female
  • Contraceptives, Oral, Synthetic
  • Drug Combinations
  • Estradiol Congeners
  • Lipids
  • Lipoproteins, HDL
  • Lipoproteins, LDL
  • Ethinyl Estradiol
  • Levonorgestrel