An F-box protein, FWD1, mediates ubiquitin-dependent proteolysis of beta-catenin

EMBO J. 1999 May 4;18(9):2401-10. doi: 10.1093/emboj/18.9.2401.

Abstract

beta-catenin plays an essential role in the Wingless/Wnt signaling cascade and is a component of the cadherin cell adhesion complex. Deregulation of beta-catenin accumulation as a result of mutations in adenomatous polyposis coli (APC) tumor suppressor protein is believed to initiate colorectal neoplasia. beta-catenin levels are regulated by the ubiquitin-dependent proteolysis system and beta-catenin ubiquitination is preceded by phosphorylation of its N-terminal region by the glycogen synthase kinase-3beta (GSK-3beta)/Axin kinase complex. Here we show that FWD1 (the mouse homologue of Slimb/betaTrCP), an F-box/WD40-repeat protein, specifically formed a multi-molecular complex with beta-catenin, Axin, GSK-3beta and APC. Mutations at the signal-induced phosphorylation site of beta-catenin inhibited its association with FWD1. FWD1 facilitated ubiquitination and promoted degradation of beta-catenin, resulting in reduced cytoplasmic beta-catenin levels. In contrast, a dominant-negative mutant form of FWD1 inhibited the ubiquitination process and stabilized beta-catenin. These results suggest that the Skp1/Cullin/F-box protein FWD1 (SCFFWD1)-ubiquitin ligase complex is involved in beta-catenin ubiquitination and that FWD1 serves as an intracellular receptor for phosphorylated beta-catenin. FWD1 also links the phosphorylation machinery to the ubiquitin-proteasome pathway to ensure prompt and efficient proteolysis of beta-catenin in response to external signals. SCFFWD1 may be critical for tumor development and suppression through regulation of beta-catenin protein stability.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenomatous Polyposis Coli Protein
  • Animals
  • Axin Protein
  • Carrier Proteins / metabolism
  • Cytoskeletal Proteins / genetics
  • Cytoskeletal Proteins / metabolism*
  • GTP-Binding Proteins / genetics
  • GTP-Binding Proteins / metabolism*
  • Mice
  • Models, Biological
  • Mutation
  • Neoplasm Proteins / metabolism
  • Peptide Synthases / metabolism
  • Protein Binding
  • Proteins / isolation & purification
  • Recombinant Proteins / metabolism
  • Repressor Proteins*
  • SKP Cullin F-Box Protein Ligases
  • Trans-Activators*
  • Ubiquitins / metabolism*
  • beta Catenin
  • beta-Transducin Repeat-Containing Proteins

Substances

  • Adenomatous Polyposis Coli Protein
  • Axin Protein
  • Btrc protein, mouse
  • CTNNB1 protein, mouse
  • Carrier Proteins
  • Cytoskeletal Proteins
  • Neoplasm Proteins
  • Proteins
  • Recombinant Proteins
  • Repressor Proteins
  • Trans-Activators
  • Ubiquitins
  • beta Catenin
  • beta-Transducin Repeat-Containing Proteins
  • SKP Cullin F-Box Protein Ligases
  • GTP-Binding Proteins
  • Peptide Synthases