Increased association of glycoprotein 120-CD4 with HIV type 1 coreceptors in the presence of complex-enhanced anti-CD4 monoclonal antibodies

AIDS Res Hum Retroviruses. 1999 Jan 20;15(2):149-59. doi: 10.1089/088922299311574.

Abstract

CD4-specific monoclonal antibodies (CG1, CG7, and CG8), which bind with a 5- to 10-fold higher avidity to preformed CD4-gp120 complexes than to CD4, were previously shown to recognize newly identified conformational epitopes in the D1-CDR3 region of CD4. In the current study, these and other complex-enhanced MAbs were tested in three separate assays of HIV-1 coreceptor (CXCR4/CCR5) recruitment. In these assays, the CD4-specific MAbs CG1, -7, and -8 stabilized the association of coreceptor, gp120, and CD4 in trimolecular complexes. In contrast, the gp120-specific, complex-enhanced MAbs 48d and 17b were inhibitory. These data suggest that conformational changes in the CDR3 region of CD4-D1, induced by gp120 binding, may be involved in coreceptor association and thus play a positive role in the HIV-1 cell fusion process.

Publication types

  • Comparative Study

MeSH terms

  • Antibodies, Monoclonal / metabolism*
  • CD4 Antigens / immunology*
  • Cell Line
  • Epitopes / immunology*
  • Flow Cytometry
  • HIV Envelope Protein gp120 / immunology
  • HIV Envelope Protein gp120 / metabolism*
  • HIV-1 / immunology
  • HIV-1 / metabolism*
  • HeLa Cells
  • Humans
  • Immunoglobulin Variable Region / metabolism
  • Jurkat Cells
  • Precipitin Tests
  • Receptors, CCR5 / metabolism
  • Receptors, CXCR4 / metabolism

Substances

  • Antibodies, Monoclonal
  • CD4 Antigens
  • Epitopes
  • HIV Envelope Protein gp120
  • Immunoglobulin Variable Region
  • Receptors, CCR5
  • Receptors, CXCR4